Generic
Ethinyl Estradiol + Lynestrenol (0.05 mg)
2 brands available in the market
At a glance
Ethinyl Estradiol + Lynestrenol (0.05 mg) is a combined oral contraceptive pill used for the prevention of pregnancy.
Description
Ethinyl Estradiol + Lynestrenol (0.05 mg) is a combined oral contraceptive pill indicated for oral contraception. It is used for the prevention of pregnancy.
This pill prevents ovulation and provides contraceptive action. It thickens cervical mucus to make sperm penetration difficult and causes changes in the endometrium to prevent implantation.
Indications
- Contraception: Used as a combined oral contraceptive pill for prevention of pregnancy.
Therapeutic class
Oral Contraceptive preparations
Pharmacological class
Combined Oral Contraceptive
Pharmacology
Ethinyl Estradiol + Lynestrenol is a combined oral contraceptive pill indicated for oral contraception. It prevents ovulation and causes changes in cervical mucus and endometrium for contraceptive action.
Mechanism of action
Ethinyl Estradiol + Lynestrenol prevents ovulation by suppressing pituitary gonadotropin secretion. It also causes changes in cervical mucus and endometrium for contraceptive action.
Dosage
Adult Dose:
- 1 tablet daily for 22 days, then 6 days tablet-free break.
- Take at the same time every day.
Administration
Take 1 tablet at the same time every day. Start from the first day of menstruation from the top row of the pack. Take 22 tablets, then 6 days break. Swallow each pill whole with water if necessary.
Missed dose
If less than 12 hours late: Take as soon as remembered; effectiveness maintained. If more than 12 hours late: Effectiveness may be reduced; take 2 tablets the next day.
Side effects
Common Side Effects:
- Headache
- Nausea
- Weight gain
- Mood changes
- Breast pain
- High blood pressure
- Blood clotting in arteries
- Liver and kidney function disturbances
Precautions & warnings
Precautions:
- Caution in cardiovascular disorders, history of thrombophlebitis and thromboembolism.
- Caution in severe hypertension, severe liver disease, history of cholestatic jaundice.
- Do not use in estrogen-dependent tumors, endometrial hyperplasia, porphyria.
- Women over 35 years who smoke should avoid smoking.
Contraindications
Contraindications:
- Cardiovascular disorders (thrombophlebitis and thromboembolic processes)
- Severe hypertension
- Severe liver disease
- History of cholestatic jaundice
- Estrogen-dependent tumors
- Endometrial hyperplasia
- Undiagnosed vaginal bleeding
- Porphyria
- Pregnancy
Drug interactions
Drug Interactions:
- Ampicillin, tetracycline, barbiturates, hydantoins, primidone, carbamazepine, rifampicin: May reduce pill effectiveness.
Food interactions
Food Interactions: May be taken with or without food. Caution with alcohol.
Use in pregnancy
Use in Pregnancy: Do not use during pregnancy.
Pregnancy Category: B3 — always consult a doctor before taking during pregnancy.
Use in lactation
Use in Lactation: Not recommended during breastfeeding.
Pediatric use
Pediatric Use: Not indicated before menarche.
Geriatric use
Geriatric Use: For women aged 15-69 years (except smokers and tobacco users).
Renal / hepatic impairment
Renal Impairment: Use with caution in patients with kidney disease.
Hepatic Impairment: Use with caution in patients with liver disease; contraindicated in severe liver disease.
Overdose effects
Overdose: Overdose may cause nausea, vomiting, vaginal bleeding. No specific antidote; symptomatic treatment.
Storage conditions
Storage: Store at 2-30 degree C in a cool and dry place, protected from light. Keep out of reach of children.
Chemical structure
Ethinyl Estradiol + Lynestrenol (0.05 mg)