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At a glance

Tiemonium Methylsulphate is an anticholinergic-antispasmodic drug that reduces muscle spasm of the intestine, biliary system, bladder, and uterus. It helps relieve pain.

Indications
  • Dysentery, diarrhea, gastroenteritis
  • Biliary colic, enterocolitis, cholecystitis
  • Colonopathies, mild cystitis
  • Spasmodic dysmenorrhea
  • Visceral muscle spasm
Pharmacology

Tiemonium Methylsulphate acts as a competitive antagonist of acetylcholine and histamine and strengthens calcium bonding with phospholipids and proteins. It inhibits intracellular contractile proteins of visceral cells, inhibiting visceral spasm and pain.

Dosage

Adult Dose:

  • Tablet: 2-6 tablets (100-300 mg) daily in divided doses
  • Syrup: 3-9 teaspoonfuls daily in divided doses
  • Injection: 1 ampoule 3 times daily (slow IV/IM)
  • Suppository: 20 mg suppository 2-3 times daily (rectal)

Pediatric Dose:

  • 3 mL/kg or 6 mg/kg body weight daily in divided doses
Side effects

Side Effects:

  • Hypotension (especially with injection)
  • Tachycardia (especially with injection)
  • Visual disturbances
  • Dry mouth
Use in pregnancy

Use in Pregnancy: Animal studies show no teratogenic effects; caution due to insufficient data; consult your doctor.

Pregnancy Category: C — always consult a doctor before taking during pregnancy.

Precautions & warnings
  • Caution in prostate disorders, serious kidney/liver disease, cardiac disorders, thyroid disorders, chronic bronchitis
  • Risk of visual disturbances may make driving or using machines dangerous
Overdose effects

No overdose information available; excessive doses may increase anticholinergic effects; consult your doctor.

Storage conditions

Store in a dry place, away from light and heat; keep out of reach of children.

Tiemonium Methylsulphate — see the full informationPharmacology, precautions, pregnancy, overdose and the rest on the generic page
⚠️ This information is for educational purposes only — not a substitute for medical advice. Consult a registered physician before taking any medicine.